Peptide | Kiδ(μM) | Kiδ/Kiκ | Kiμ/Kiκ |
---|---|---|---|
1. Dmt-Tic-OH | 23,806 ± 2,697 (3) | 0.0000009 | 0.14 |
2. Dmt-Tic-NH2 | 1,943 ± 113 (3) | 0.0006 | 0.14 |
3. Dmt-d-Tic-OH | 9,863 ± 2,621 (3) | 0.0014 | 0.02 |
4. Dmt-d-Tic-NH2 | 5,291 ± 105 (3) | 0.011 | 0.0007 |
5. Dmt-Tic-CH2OH | 1,107 ± 158 (4) | 0.0004 | 0.14 |
6. Tyr-Tic-OH | >60,000 | − | — |
11. Dmt-Tic-Ala-OH | >50,000 (3) | <0.000006 | 0.12 |
12. Dmt-Tic-Ala-NH2 | 8,694 ± 1,254 (5) | 0.000028 | 0.005 |
13. Dmt-d-Tic-Ala-OH | 9,752 ± 2,418 (3) | 0.009 | 0.008 |
14. Dmt-d-Tic-Ala-NH2 | 7,087 ± 2,181 (3) | 0.0007 | 0.0008 |
15. Tyr-Tic-Ala-OH | >60,000 | − | — |
16. Tyr-Tic-Ala-NH2 | >60,000 | − | — |